四优青年 国家优秀青年科学基金获得者

丁克

职务:

暨南大学药学院院长

职称:

教授

研究工作:

1、基于功能蛋白结构的小分子调节剂的设计与合成。

2、表观遗传学小分子调控与干细胞化学生物学。

代表性学术论文:

1、Shaohua Chang,Lianwen Zhang,Shilin Xu,Jinfeng Luo,Xiaoyun Lu,Zhang Zhang,Tianfeng Xu,Yingxue Liu,Zhengchao Tu,Yong Xu,Xiaomei Ren,Meiyu Geng,Jian Ding,Duanqing Pei and Ke Ding.* Design,Synthesis and Biological Evaluation of Novel Conformationally Constrained Inhibitors Targeting Epidermal Growth Factor Receptor Threonine790 ® Methionine790 mutant.J.Med.Chem.2012,55,2711-2723.

2、Huimin Cheng,Junting Wan,Meng-I Lin,Yingxue Liu,Xiaoyun,Lu,Jinsong Liu,Yong Xu Jianxin Chen,Zhengchao Tu,Yih-Shyun E.Cheng,and Ke Ding*.Design,synthesis and in vitro biological evaluation of 1H-1,2,3-triazole-4-carboxamide derivatives as new anti-influenza A agents targeting virus nucleoprotein.J.Med.Chem.2012,55 (5),2144–2153.

3、Yupeng Li,Mengjie Shen,Zhang Zhang,Jinfeng Luo,Xiaofen Pan,Xiaoyun Lu,Huoyou Long,Donghai Wen,Fengxiang Zhang,Fang Leng,Yingjun Li,Zhengchao Tu,Xiaomei Ren,and Ke Ding *.Design,Synthesis,and Biological Evaluation of 3-(1H-1,2,3-Triazol-1-yl)benzamide Derivatives as Potent Pan Bcr-Abl Inhibitors Including the Threonine315→Isoleucine315 Mutant.J.Med.Chem.,2012,DOI: 10.1021/jm301188x

4、Shilin Xu,Lianwen Zhang,Shaohua Chang,Jinfeng Luo,Xiaoyun Lu,Zhengchao Tu,Yingxue Liu,Zhang zhang,Yong Xu,Xiaomei Ren and Ke Ding.* Design,synthesis and biological evaluation of new molecules inhibiting epidermal growth factor receptor threonine790→ methionine790 mutant.Med.Chem.Commun.,2012,3,1155-1159.

5、Lijie Peng,Xuefei Gao,Lei Duan,Xiaomei Ren,Donghai Wu,and Ke Ding.* Identification of Pyrido[1,2-α]pyrimidine-4-ones as New Molecules Improving the Transcriptional Functions of Estrogen-Related Receptor α.J.Med.Chem.2011,54,7729–7733.

获奖及个人荣誉:

1、2007 中国科学院“百人计划” 2008

2、广州市优秀专家 2007-2008年度

3、中科院广州教育基地优秀研究生导师 2010

4、广东省丁颖科技奖 2011-2012年度

5、中科院广州教育基地优秀研究生导师 2012

6、中国科学院“百人计划”终期评估优秀


联系方式:

Email: ding_ke@gibh.ac.cn